Last updated: 06/23/2026 18:00:17

A study to evaluate the safety,tolerability, pharmacokinetics and clinical activity of Mocertatug Rezetecan for injection in participants with advanced solid tumors (BEHOLD-1)

GSK study ID
222730
Clinicaltrials.gov ID
EudraCT ID
Not applicable
EU CT Number
Trial status
Recruiting
Recruiting
Overview
Eligibility
Locations
Study documents
Results summary
Plain language summaries
Additional information

Trial overview

Official title: A Phase 1 Clinical Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Clinical Activity of Mocertatug Rezetecan for Injection in Subjects with Advanced Solid Tumors
Trial description: The goal of this study is to assess the safety and tolerability of Mocertatug Rezetecan . The study will also see how the levels of Mo-Rez change over time at different dose amount
Primary purpose:
Treatment
Trial design:
Sequential Assignment
Masking:
None (Open Label)
Allocation:
Randomized
Primary outcomes:

Part 1: Number of participants with dose limiting toxicity (DLT)

Timeframe: Up to 21 days

Part 2-Confirmed Objective Response Rate (ORR) assessed by investigator

Timeframe: Up to approximately 28 months

Secondary outcomes:

Part 1 and 2: Maximum observed concentration (Cmax) of Mocertatug Rezetecan and its components: conjugated antibody, total antibody, and small molecule toxin

Timeframe: Up to approximately 31 months

Part 1 and 2: Time to reach Cmax (Tmax) of Mocertatug Rezetecan and its components: conjugated antibody, total antibody, and small molecule toxin

Timeframe: Up to approximately 31 months

Part 1 and 2: Area under the concentration-time curve (AUC) of Mocertatug Rezetecan and its components: conjugated antibody, total antibody, and small molecule toxin

Timeframe: Up to approximately 31 months

Part 1- Confirmed Objective Response Rate assessed by investigator

Timeframe: Up to approximately 31 months

Part 1 and 2: Duration of response (DoR) assessed by investigator

Timeframe: Up to approximately 31 months

Part 1 and 2: Progression-free survival (PFS) assessed by investigator

Timeframe: Up to approximately 31 months

Part 1 and 2: Number of participants with treatment-emergent Anti-drug antibodies (ADA) / Neutralizing antibody (NAb)

Timeframe: Up to approximately 31 months

Part 1 and 2: Titers of ADA to Mocertatug Rezetecan

Timeframe: Up to approximately 31 months

Part 1 and 2: Number of participants with Adverse Events (AEs), Serious Adverse Events (SAEs) and Adverse Events of Special Interest (AESIs)

Timeframe: Up to approximately 31 months

Part 1 and 2: Change from baseline in body temperature (degree Celsius)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in respiratory rate (breaths per minute)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in pulse rate (beats per minute)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in blood pressure [millimetres of mercury (mmHg)]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in weight [kilogram (kg)]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in white blood cell count (cells per microliter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in hemoglobin (grams per deciliter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from Baseline in Platelet count (cells per microliter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from Baseline in Red Blood Cell Count (RBC) (million cells per microliter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from Baseline in haematocrit (Proportion of red blood cells in blood)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from Baseline in Neutrophils, Lymphocytes, Monocytes, Eosinophils, Basophils (giga cells per litre)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from Baseline in Glucose (fasting), Blood Urea Nitrogen (BUN), Creatinine, Sodium, Potassium, Calcium, Chloride, Magnesium Direct Bilirubin and Total Bilirubin (milligrams per decilitre)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from Baseline in AST/SGOT, ALT/ SGPT, ALP and CPK (International Units per litre)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Total Protein and Albumin (Grams per deciliter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Amylase and Lipase (Units per liter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Estimated glomerular filtration rate (eGFR) (milliliter per minute)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Prothrombin Time (PT), Partial thromboplastin time (PTT) or Activated Partial Thromboplastin Time (aPTT) (seconds)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in liver panel parameter: International Normalized Ratio (INR)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in routine urine tests: Leukocyte esterase

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in routine urine tests: Occult blood (10^9 Cells Per Liter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in routine urine tests: potential of hydrogen (pH) value

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in routine urine tests: Protein and bilirubin (Grams Per Liter)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change From Baseline in routine urine tests: Specific Gravity (Ratio)

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in CA-125 tumor marker among ovarian cancer participants [units per milliliter (U/mL)]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Thyroid stimulating hormone (TSH) [microunits per milliliter (µU/mL)]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in free thyroxine (T4) [nanograms per deciliter (ng/dL)]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Electrocardiogram (ECG) readings [milliseconds (msec)]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Left ventricular ejection fraction (LVEF) [Percentage]

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 1 and 2: Change from baseline in Eastern Cooperative Oncology Group Performance Scale (ECOG PS) score

Timeframe: Baseline (Day -1) and up to approximately 31 months

Part 2: Overall Survival (OS)

Timeframe: Up to approximately 31 months

Part 2-Confirmed Objective Response Rate (ORR) assessed by BICR

Timeframe: Up to approximately 31 months

Part 2: Duration of response (DoR) assessed by BICR

Timeframe: Up to approximately 31 months

Part 2: Progression-free survival (PFS) assessed by BICR

Timeframe: Up to approximately 31 months

Interventions:
Drug: Mocertatug rezetecan
Enrollment:
675
Primary completion date:
2027-22-09
Observational study model:
Not applicable
Time perspective:
Not applicable
Clinical publications:
Not applicable
Medical condition
Solid Tumors, Neoplasms
Product
GSK5733584
Collaborators
Not applicable
Study date(s)
July 2024 to December 2029
Type
Interventional
Phase
1

Participation criteria

Sex
Female & Male
Age
18+ years
Accepts healthy volunteers
No
  • Males or females aged 18 years or older (≥18 years).
  • Participants with pathologically confirmed advanced solid tumor (who have failed or are intolerant to standard of care.
  • Have received any B7-H4-targeted therapy
  • Have received any of cytotoxic chemotherapy drugs, anti-tumor traditional Chinese medicines or other anti-tumor drugs within 28 days prior to the first dose of study drug; or need to continue these drugs during the study.

Trial location(s)

Location
Status
Contact us
Contact us
Location
GSK Investigational Site
Leuven, Belgium, 3000
27.9 miles (44.6 km) away from your location
Status
Recruiting

Study documents

No study documents available.

Results overview

Study Results yet to be posted

Recruitment status
Recruiting
Actual primary completion date
Not applicable
Actual study completion date
Not applicable

Plain language summaries

Plain language summaries of clinical trial results for Phase 2-4 clinical trials that were initiated on or after January 2022 will be posted by GSK within one year following study completion.

Additional information about the trial

Additional information
Not applicable
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